Novel Benzamide-Based Histamine H3 Receptor Antagonists: The Identification of Two Candidates for Clinical Development-Reference-Cited by-同舟云学术

Novel Benzamide-Based Histamine H3 Receptor Antagonists: The Identification of Two Candidates for Clinical Development

Published:2015-03-16 Issue:4 Volume:6 Page:450-454
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Letavic Michael A.¹,Aluisio Leah¹,Apodaca Richard¹,Bajpai Manoj¹,Barbier Ann J.¹,Bonneville Anne¹,Bonaventure Pascal¹,Carruthers Nicholas I.¹,Dugovic Christine¹,Fraser Ian C.¹,Kramer Michelle L.¹,Lord Brian¹,Lovenberg Timothy W.¹,Li Lilian Y.¹,Ly Kiev S.¹,Mcallister Heather¹,Mani Neelakandha S.¹,Morton Kirsten L.¹,Ndifor Anthony¹,Nepomuceno S. Diane¹,Pandit Chennagiri R.¹,Sands Steven B.¹,Shah Chandra R.¹,Shelton Jonathan E.¹,Snook Sandra S.¹,Swanson Devin M.¹,Xiao Wei¹

Affiliation:

1. Janssen Pharmaceutical Company, a division of Johnson & Johnson Pharmaceutical Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml5005156

Reference14 articles.

1. The histamine H3receptor: an attractive target for the treatment of cognitive disorders

2. The histamine H3 receptor as a therapeutic drug target for CNS disorders

3. Histamine H3 Receptor Antagonists Go to Clinics

4. Histamine H3 Antagonists as Wake-Promoting and Pro-Cognitive Agents

5. Histamine H3 Receptor Function and Ligands: Recent Developments

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