Development of a Scalable and Safe Procedure for the Production of (3R)-3-(2,3-Dihydro-1-benzofuran-5-yl)-1,2,3,4-tetrahydro-9H-pyrrolo[3,4-b]- quinolin-9-one, an Intermediate in the Synthesis of PDE-V Inhibitors RWJ387273 (R301249) and RWJ444772 (R290629)-Reference-Cited by-同舟云学术

Development of a Scalable and Safe Procedure for the Production of (3R)-3-(2,3-Dihydro-1-benzofuran-5-yl)-1,2,3,4-tetrahydro-9H-pyrrolo[3,4-b]- quinolin-9-one, an Intermediate in the Synthesis of PDE-V Inhibitors RWJ387273 (R301249) and RWJ444772 (R290629)

Published:2006-07-12 Issue:6 Volume:10 Page:1275-1281
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Willemsens Bert¹,Vervest Ivan¹,Ormerod Dominic¹,Aelterman Wim¹,Fannes Christine¹,Mertens Narda¹,Markó István E.¹,Lemaire Sebastien¹

Affiliation:

1. Chemical Development, Johnson & Johnson Pharmaceutical Research & Development, Turnhoutseweg 30, 2340 Beerse, Belgium, and Université Catholique de Louvain, Laboratoire de Chimie Organique, Place Louis Pasteur, 1, 1348 Louvain-la-Neuve, Belgium

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op060099f

Reference10 articles.

1. Sui, Z.; Macielag, M. J.; Guan, J.; Jiang, W.; Lanter, J. C. PCT Int. Appl.2001 WO0187882.

2. Reaktionen an Indolderivaten, XIII. Chinolon-Derivate durch Autoxydation

3. Reaktionen an Indolderivaten, XVII. Die biogenetisch orientierte Totalsynthese von DL‐Camptothecin und 7‐Chlor‐camptothecin

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