Discovery of N-Hydroxyindole-Based Inhibitors of Human Lactate Dehydrogenase Isoform A (LDH-A) as Starvation Agents against Cancer Cells-Reference-Cited by-同舟云学术

Discovery of N-Hydroxyindole-Based Inhibitors of Human Lactate Dehydrogenase Isoform A (LDH-A) as Starvation Agents against Cancer Cells

Published:2011-02-18 Issue:6 Volume:54 Page:1599-1612
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Granchi Carlotta,Roy Sarabindu,Giacomelli Chiara,Macchia Marco,Tuccinardi Tiziano,Martinelli Adriano,Lanza Mario,Betti Laura,Giannaccini Gino,Lucacchini Antonio,Funel Nicola¹,León Leticia G.²³,Giovannetti Elisa³,Peters Godefridus J.³,Palchaudhuri Rahul⁴,Calvaresi Emilia C.⁴,Hergenrother Paul J.⁴,Minutolo Filippo

Affiliation:

1. Dipartimento di Chirurgia (Anatomia Patologica), Università di Pisa, Via Roma 57, 56126 Pisa, Italy

2. Institudo Universitario de Bio-Organica “Antonio Gonzales”, Universidad de La Laguna, Avda. Astrofisico F. Sánchez 2, La Laguna, 38206-Tenerife, Spain

3. Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands

4. Department of Chemistry, University of Illinois, 600 S. Mathews Avenue, Urbana, Illinois 61801, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm101007q

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