Indole-3-acetic Acid Antagonists of the Prostaglandin D2 Receptor CRTH2-Reference-Cited by-同舟云学术

Indole-3-acetic Acid Antagonists of the Prostaglandin D2 Receptor CRTH2

Published:2005-09-10 Issue:20 Volume:48 Page:6174-6177
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Armer Richard E.¹,Ashton Mark R.¹,Boyd Edward A.¹,Brennan Chris J.¹,Brookfield Frederick A.¹,Gazi Lucien¹,Gyles Shân L.¹,Hay Philip A.¹,Hunter Michael G.¹,Middlemiss David¹,Whittaker Mark¹,Xue Luzheng¹,Pettipher Roy¹

Affiliation:

1. Oxagen Ltd., 91 Milton Park, Abingdon, Oxfordshire, OX14 4RY, U.K., Evotec OAI, 151 Milton Park, Abingdon, Oxfordshire, OX14 4SD, U.K., and XaviaPharm, 61 Thorley Hill, Bishop's Stortford, Hertfordshire, CM23 3NF, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050519b

Reference26 articles.

1. The Bronchoconstrictor Effect of Inhaled Prostaglandin D2 in Normal and Asthmatic Men

2. Prostaglandin D2 causes accumulation of eosinophils in the lumen of the dog trachea

3. Prostaglandin D2-Induced Eosinophilic Airway Inflammation Is Mediated by CRTH2 Receptor

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