[11C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor-Reference-Cited by-同舟云学术

[11C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor

Published:2013-07-18 Issue:9 Volume:4 Page:863-868
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Bell Ian M.¹,Gallicchio Steven N.¹,Stump Craig A.¹,Bruno Joseph G.¹,Fan Hong¹,Gantert Liza T.¹,Hostetler Eric D.¹,Kemmerer Amanda L.¹,McWherter Melody¹,Moore Eric L.¹,Mosser Scott D.¹,Purcell Mona L.¹,Riffel Kerry¹,Salvatore Christopher A.¹,Sanabria-Bohórquez Sandra¹,Staas Donnette D.¹,White Rebecca B.¹,Williams Mangay¹,Zartman C. Blair¹,Cook Jacquelynn J.¹,Hargreaves Richard J.¹,Kane Stefanie A.¹,Graham Samuel L.¹,Selnick Harold G.¹

Affiliation:

1. Departments of †Medicinal Chemistry, ‡Pain & Migraine, §Imaging, ∥In Vitro Pharmacology, ⊥Neuroscience & Ophthalmology, and #Pharmacokinetics Pharmacodynamics & Drug Metabolism, Merck Research Laboratories, West Point, Pennsylvania 19486, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml400199p

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4. Calcitonin Gene–Related Peptide Receptor Antagonist BIBN 4096 BS for the Acute Treatment of Migraine

5. Efficacy and tolerability of MK-0974 (telcagepant), a new oral antagonist of calcitonin gene-related peptide receptor, compared with zolmitriptan for acute migraine: a randomised, placebo-controlled, parallel-treatment trial

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