Identification of Selective, Nonpeptidic Nitrile Inhibitors of Cathepsin S Using the Substrate Activity Screening Method-Reference-Cited by-同舟云学术

Identification of Selective, Nonpeptidic Nitrile Inhibitors of Cathepsin S Using the Substrate Activity Screening Method

Published:2006-09-12 Issue:21 Volume:49 Page:6298-6307
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Patterson Andrew W.¹,Wood Warren J. L.¹,Hornsby Michael¹,Lesley Scott¹,Spraggon Glen¹,Ellman Jonathan A.¹

Affiliation:

1. Department of Chemistry, University of California, Berkeley, California 94720, and Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060701s

Reference35 articles.

1. Rapid Identification of Potent Nonpeptidic Serine Protease Inhibitors

2. A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

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