Discovery of a Potent, Non-peptide Bradykinin B1 Receptor Antagonist-Reference-Cited by-同舟云学术

Discovery of a Potent, Non-peptide Bradykinin B1 Receptor Antagonist

Published:2003-05-31 Issue:25 Volume:125 Page:7516-7517
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Su Dai-Shi¹,Markowitz M. Kristine¹,DiPardo Robert M.¹,Murphy Kathy L.¹,Harrell C. Meacham¹,O'Malley Stacy S.¹,Ransom Richard W.¹,Chang Raymond S. L.¹,Ha Sookhee¹,Hess Fred J.¹,Pettibone Douglas J.¹,Mason Glenn S.¹,Boyce Susan¹,Freidinger Roger M.¹,Bock Mark G.¹

Affiliation:

1. Departments of Medicinal Chemistry and Neuroscience, Merck Research Laboratories, West Point, Pennsylvania 19486, and Neuroscience Research Centre, Merck Research Laboratories, Terlings Park, Harlow, Essex, CM20 2QR, England

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja0353457

Reference7 articles.

1. Hypoalgesia and altered inflammatory responses in mice lacking kinin B1 receptors

2. Crystal Structure of Rhodopsin: A G Protein-Coupled Receptor

3. A Single Position in the Third Transmembrane Domains of the Human B1 and B2 Bradykinin Receptors Is Adjacent to and Discriminates between the C-terminal Residues of Subtype-selective Ligands

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