Novel 5-HT7 Receptor Inverse Agonists. Synthesis and Molecular Modeling of Arylpiperazine- and 1,2,3,4-Tetrahydroisoquinoline-Based Arylsulfonamides-Reference-Cited by-同舟云学术

Novel 5-HT7 Receptor Inverse Agonists. Synthesis and Molecular Modeling of Arylpiperazine- and 1,2,3,4-Tetrahydroisoquinoline-Based Arylsulfonamides

Published:2004-09-23 Issue:22 Volume:47 Page:5451-5466
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Vermeulen Erik S.¹,van Smeden Marjan¹,Schmidt Anne W.¹,Sprouse Jeffrey S.¹,Wikström Håkan V.¹,Grol Cor J.¹

Affiliation:

1. Department of Medicinal Chemistry, Center for Pharmacy, State University of Groningen, A. Deusinglaan 1, NL-9713 AV Groningen, The Netherlands, and Pfizer Global R & D, Department of Neuroscience, MS 8220-4178, Groton, Connecticut 06340

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049743b

Reference48 articles.

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5. An alpha-carbon template for the transmembrane helices in the rhodopsin family of G-protein-coupled receptors 1 1Edited by R. Huber

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