Disrupting the Constitutive, Homodimeric Protein–Protein Interface in CK2β Using a Biophysical Fragment-Based Approach
Author:
Affiliation:
1. Department of Chemistry, University of Cambridge, Lensfield Road, Cambridge, CB2 1EW, United Kingdom
Funder
Agency for Science, Technology and Research
Wellcome Trust
Publisher
American Chemical Society (ACS)
Subject
Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis
Link
http://pubs.acs.org/doi/pdf/10.1021/jacs.6b07440
Reference60 articles.
1. Protein kinase CK2: structure, regulation and role in cellular decisions of life and death
2. Crystal structure of human protein kinase CK2: insights into basic properties of the CK2 holoenzyme
3. New Protein Kinase CK2 Inhibitors: Jumping out of the Catalytic Box
4. Structure-based design of small peptide inhibitors of protein kinase CK2 subunit interaction
5. Identification of chemical inhibitors of protein-kinase CK2 subunit interaction
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