Potent and Fully Noncompetitive Peptidomimetic Inhibitor of Multidrug Resistance P-Glycoprotein-Reference-Cited by-同舟云学术

Potent and Fully Noncompetitive Peptidomimetic Inhibitor of Multidrug Resistance P-Glycoprotein

Published:2010-08-23 Issue:18 Volume:53 Page:6720-6729
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Arnaud Ophélie¹,Koubeissi Ali²,Ettouati Laurent²,Terreux Raphaël¹,Alamé Ghina³,Grenot Catherine³,Dumontet Charles⁴,Di Pietro Attilio¹,Paris Joëlle²,Falson Pierre¹

Affiliation:

1. Laboratoire des Protéines de Résistance aux Agents Chimiothérapeutiques, Equipe Labellisée Ligue 2009, Institut de Biologie et Chimie des Protéines, UMR 5086 CNRS, Université Lyon 1, IFR 128 BioSciences Gerland Lyon-Sud, F-69367 Lyon, France

2. EA 3741 Écosystèmes et Molécules Bioactives, Institut des Sciences Pharmaceutiques et Biologiques, Université de Lyon, Université Claude Bernard Lyon 1, F-69373 Lyon, France

3. Université de Lyon, Université Claude Bernard Lyon 1, INSERM, U863, F-69373 Lyon, France

4. Laboratoire de Cytologie Analytique, Faculté de Médecine, Université de Lyon, Université Claude Bernard Lyon 1, INSERM U590, F-69373 Lyon, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100839w

Reference39 articles.

1. The human ATP-binding cassette (ABC) transporter superfamily

2. Breast Cancer Resistance Protein (BCRP/ABCG2) Induces Cellular Resistance to HIV-1 Nucleoside Reverse Transcriptase Inhibitors

3. Modulation of human BCRP (ABCG2) activity by anti-HIV drugs

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