New Non-Peptide Endothelin-A Receptor Antagonists: Synthesis, Biological Properties, and Structure−Activity Relationships of 5-(Dimethylamino)-N-pyridyl-, -N-pyrimidinyl-, -N-pyridazinyl-, and -N-pyrazinyl-1-naphthalenesulfonamides-Reference-Cited by-同舟云学术

New Non-Peptide Endothelin-A Receptor Antagonists: Synthesis, Biological Properties, and Structure−Activity Relationships of 5-(Dimethylamino)-N-pyridyl-, -N-pyrimidinyl-, -N-pyridazinyl-, and -N-pyrazinyl-1-naphthalenesulfonamides

Published:1997-03-01 Issue:6 Volume:40 Page:996-1004
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bradbury Robert H.¹,Bath Colin¹,Butlin Roger J.¹,Dennis Michael¹,Heys Christine¹,Hunt Sarah J.¹,James Roger¹,Mortlock Andrew A.¹,Sumner Neil F.¹,Tang Eric K.¹,Telford Berwick¹,Whiting Elaine¹,Wilson Campbell¹

Affiliation:

1. Cardiovascular and Musculoskeletal Department, ZENECA Pharmaceuticals, Mereside, Alderley Park, Macclesfield, Cheshire SK10 4TG, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9604585

Reference55 articles.

1. A novel potent vasoconstrictor peptide produced by vascular endothelial cells

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