Synthesis of Chiral TFA-Protected α-Amino Aryl-Ketone Derivatives with Friedel–Crafts Acylation of α-Amino Acid N-Hydroxysuccinimide Ester-Reference-Cited by-同舟云学术

Synthesis of Chiral TFA-Protected α-Amino Aryl-Ketone Derivatives with Friedel–Crafts Acylation of α-Amino Acid N-Hydroxysuccinimide Ester

Published:2017-10-17 Issue:10 Volume:22 Page:1748
ISSN:1420-3049
Container-title:Molecules
language:en
Short-container-title:Molecules

Author:

Tachrim Zetryana,Oida Kazuhiro,Ikemoto Haruka,Ohashi Fumina,Kurokawa Natsumi,Hayashi Kento,Shikanai Mami,Sakihama Yasuko,Hashidoko Yasuyuki,Hashimoto Makoto

Publisher

MDPI AG

Subject

Chemistry (miscellaneous),Analytical Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Molecular Medicine,Drug Discovery,Pharmaceutical Science

Link

http://www.mdpi.com/1420-3049/22/10/1748/pdf

Reference26 articles.

1. Facile Approach to Enantiomerically Pure α-Amino Ketones by Friedel−Crafts Aminoacylation and Their Conversion into Peptidyl Ketones

2. Friedel-Crafts acylation with N-(trifluoroacetyl)-.alpha.-amino acid chlorides. Application to the preparation of .beta.-arylalkylamines and 3-substituted 1,2,3,4-tetrahydroisoquinolines

3. Friedel–Crafts and Related Reactions;Olah,1963

4. Friedel–Crafts and Related Reactions;Olah,1964

5. Trifluoromethanesulfonic Acid as Acylation Catalyst: Special Feature for C- and/or O-Acylation Reactions

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