Exploring the Metabolism of (+)-[18F]Flubatine In Vitro and In Vivo: LC-MS/MS Aided Identification of Radiometabolites in a Clinical PET Study †-Reference-Cited by-同舟云学术

Exploring the Metabolism of (+)-[18F]Flubatine In Vitro and In Vivo: LC-MS/MS Aided Identification of Radiometabolites in a Clinical PET Study †

Published:2018-02-20 Issue:2 Volume:23 Page:464
ISSN:1420-3049
Container-title:Molecules
language:en
Short-container-title:Molecules

Author:

Ludwig Friedrich-Alexander,Fischer Steffen,Smits René,Deuther-Conrad Winnie,Hoepping Alexander,Tiepolt Solveig,Patt Marianne,Sabri Osama,Brust Peter^ORCID

Publisher

MDPI AG

Subject

Chemistry (miscellaneous),Analytical Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Molecular Medicine,Drug Discovery,Pharmaceutical Science

Link

http://www.mdpi.com/1420-3049/23/2/464/pdf

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4. LC-MS Supported Studies on the in Vitro Metabolism of both Enantiomers of Flubatine and the in Vivo Metabolism of (+)-[18F]Flubatine—A Positron Emission Tomography Radioligand for Imaging α4β2 Nicotinic Acetylcholine Receptors

5. In vivo measurement of nicotinic acetylcholine receptors with [18F]norchloro-fluoro-homoepibatidine

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