Advancements in Non-Addictive Analgesic Diterpenoid Alkaloid Lappaconitine: A Review

Author:

Zhang Wen12,Mi Shujuan1,He Xinxin1,Cui Jiajia12,Zhi Kangkang12,Zhang Ji12

Affiliation:

1. College of Life Science, Northwest Normal University, Lanzhou 730070, China

2. Institute of New Rural Development, Northwest Normal University, Lanzhou 730070, China

Abstract

The perennial herb Aconitum sinomontanum Nakai (Ranunculaceae) has been utilized as a traditional oriental medicine in China for numerous years. The principal pharmacological constituent of A. sinomontanum, lappaconitine (LA), exhibits analgesic, anti-inflammatory, anti-tumor, anti-arrhythmic, and anti-epileptic activities. Due to its potent efficacy and non-addictive nature, LA is widely utilized in the management of cancer pain and postoperative analgesia. This review encompasses the research advancements pertaining to LA including extraction methods, separation techniques, pharmacological properties, chemical modifications, and clinical applications. Additionally, it offers insights into the potential applications and current challenges associated with LA to facilitate future research endeavors.

Funder

Projects for Science and Technology Specialist of Gansu Province

Innovation and Entrepreneurship Talent Project of Lanzhou

Enhancement Plan for Youth Teacher Research Ability of Northwest Normal University

Publisher

MDPI AG

Reference102 articles.

1. Traditional processing, uses, phytochemistry, pharmacology and toxicology of Aconitum sinomontanum Nakai: A comprehensive review;Zhang;J. Ethnopharmacol.,2022

2. Effect of lappaconitine on neuropathic pain mediated by P2X3 receptor in rat dorsal root ganglion;Ou;Neurochem. Int.,2011

3. Study of analgesic and anti-inflammatory effects of lappaconitine gelata;Wang;Chin. J. Nat. Med.,2009

4. Lappaconitine: Influence of Halogen Substituent on the Antiarrhythmic Activity;Bryzgalov;Cardiovasc. Hematol. Agents Med. Chem.,2013

5. Epilepsy-related voltage-gated sodium channelopathies: A review;Menezes;Front. Pharmacol.,2020

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3