Targeting Estrogen Receptor-α Reduces Adrenocortical Cancer (ACC) Cell Growthin Vitroandin Vivo: Potential Therapeutic Role of Selective Estrogen Receptor Modulators (SERMs) for ACC Treatment

Author:

Sirianni Rosa1,Zolea Fabiana1,Chimento Adele1,Ruggiero Carmen1,Cerquetti Lidia2,Fallo Francesco3,Pilon Catia3,Arnaldi Giorgio4,Carpinelli Giulia5,Stigliano Antonio2,Pezzi Vincenzo1

Affiliation:

1. Department of Pharmaco-Biology (R.S., F.Z., A.C., C.R., V.P.), University of Calabria, 87036 Arcavacata di Rende (CS), Italy

2. Department of Clinical and Molecular Medicine (L.C., A.S.), Sant'Andrea Hospital, Sapienza University of Rome, 1035-00189 Rome, Italy

3. Department of Medical and Surgical Sciences (F.F., C.P.), University of Padova, 35128 Padova, Italy

4. Division of Endocrinology (G.A.), University of Ancona, 60020 Ancona, Italy;

5. Department of Cell Biology and Neurosciences (G.C.), Istituto Superiore di Sanità, 00161 Rome, Italy

Publisher

The Endocrine Society

Subject

Biochemistry (medical),Clinical Biochemistry,Endocrinology,Biochemistry,Endocrinology, Diabetes and Metabolism

Reference57 articles.

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2. Adrenocortical carcinoma: clinical, morphologic, and molecular characterization.;Stojadinovic;J Clin Oncol,2002

3. Metabolism and covalent binding of 1-(o-chlorophenyl)-1-(p-chlorophenyl)-2,2-dichloroethane (o,p,′-DDD). Correlation between adrenocorticolytic activity and metabolic activation by adrenocortical mitochondria.;Martz;Drug Metab Dispos,1980

4. Loss of heterozygosity of 17p13, with possible involvement of ACADVL and ALOX15B, in the pathogenesis of adrenocortical tumors.;Soon;Ann Surg,2008

5. molecular classification and prognostication of adrenocortical tumors by transcriptome profiling.;Giordano;Clin Cancer Res,2009

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