Inhibition of pyruvate dehydrogenase kinase by halogenated acetophenones
Author:
Publisher
Wiley
Subject
Drug Discovery
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4. Synthesis, biological evaluation and structure-activity relationship of novel dichloroacetophenones targeting pyruvate dehydrogenase kinases with potent anticancer activity;European Journal of Medicinal Chemistry;2021-03
5. High-throughput screening of novel pyruvate dehydrogenase kinases inhibitors and biological evaluation of their in vitro and in vivo antiproliferative activity;European Journal of Medicinal Chemistry;2019-02
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