Structural and ITC Characterization of Peptide‐Protein Binding: Thermodynamic Consequences of Cyclization Constraints, a Case Study on Vascular Endothelial Growth Factor Ligands-Reference-Cited by-同舟云学术

Structural and ITC Characterization of Peptide‐Protein Binding: Thermodynamic Consequences of Cyclization Constraints, a Case Study on Vascular Endothelial Growth Factor Ligands

Published:2022-07-07 Issue:48 Volume:28 Page:
ISSN:0947-6539
Container-title:Chemistry – A European Journal
language:en
Short-container-title:Chemistry A European J

Author:

Gaucher Jean‐François¹^ORCID,Reille‐Seroussi Marie²,Broussy Sylvain²^ORCID

Affiliation:

1. CiTCoM UMR CNRS 8038 Université Paris Cité, Faculté de Santé, UFR de Pharmacie 4 av. de l'Observatoire 75006 Paris France

2. CitCoM UMR CNRS 8038 U1268 INSERM Université Paris Cité, Faculté de Santé, UFR de Pharmacie 4 av. de l'Observatoire 75006 Paris France

Funder

Université de Paris

Publisher

Wiley

Subject

General Chemistry,Catalysis,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/chem.202200465

Reference62 articles.

2. Conformational constraint in protein ligand design and the inconsistency of binding entropy

3. Thermodynamic and Structural Effects of Conformational Constraints in Protein−Ligand Interactions. Entropic Paradoxy Associated with Ligand Preorganization

4. Stabilizing the Pro-Apoptotic BimBH3 Helix (BimSAHB) Does Not Necessarily Enhance Affinity or Biological Activity

5. Entropy-Enthalpy Compensation: Role and Ramifications in Biomolecular Ligand Recognition and Design

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