A Series of Thiadiazolyl‐Benzenesulfonamides Incorporating an Aromatic Tail as Isoform‐Selective, Potent Carbonic Anhydrase II/XII Inhibitors-Reference-Cited by-同舟云学术

A Series of Thiadiazolyl‐Benzenesulfonamides Incorporating an Aromatic Tail as Isoform‐Selective, Potent Carbonic Anhydrase II/XII Inhibitors

Published:2022-03-09 Issue:10 Volume:17 Page:
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Banoglu Erden¹^ORCID,Ercanlı Taner¹,Gür Maz Tuğçe¹,Vullo Daniela²,Bonardi Alessandro²³,Gratteri Paola³,Supuran Claudiu T.²

Affiliation:

1. Department of Pharmaceutical Chemistry Faculty of Pharmacy Gazi University Taç Sok. No:3 Yenimahalle 06560 Ankara Turkey

2. Department of NEUROFARBA Section of Pharmaceutical and Nutraceutical Sciences University of Florence Polo Scientifico, Via Ugo Schiff 6 50019 Sesto Fiorentino Firenze Italy

3. Department of NEUROFARBA Section of Pharmaceutical and Nutraceutical Sciences Laboratory of Molecular Modeling Cheminformatics & QSAR University of Florence Polo Scientifico, Via U. Schiff 6 50019 Sesto Fiorentino Firenze Italy

Funder

Gazi Üniversitesi

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202200056

Reference27 articles.

1. Structure and function of carbonic anhydrases

2. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

4. Carbonic anhydrase inhibitors: Cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides

5. Carbonic anhydrase inhibitors

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