Recent Advances in Dual BRD4‐Kinase Inhibitors Based on Polypharmacology-Reference-Cited by-同舟云学术

Recent Advances in Dual BRD4‐Kinase Inhibitors Based on Polypharmacology

Published:2022-02-22 Issue:6 Volume:17 Page:
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Chen Li¹^ORCID,Liu Zhao‐Peng¹^ORCID,Li Xun²

Affiliation:

1. Department of Medicinal Chemistry Key Laboratory of Chemical Biology (Ministry of Education) School of Pharmaceutical Sciences Cheeloo College of Medicine Shandong University No 44, West Wenhua Road Ji'nan 250012 China

2. Institute of Materia Medica Shandong First Medical University & Shandong Academy of Medical Sciences No 6699, Qingdao Road Ji'nan 250117 China

Funder

Natural Science Foundation of Shandong Province

Ministry of Public Security of the People's Republic of China

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.202100731

Reference131 articles.

1. Disrupting Acetyl-Lysine Recognition: Progress in the Development of Bromodomain Inhibitors

2. Epigenetic protein families: a new frontier for drug discovery

4. The bromodomain: a conserved sequence found in human,Drosophilaand yeast proteins

5. brahma: A regulator of Drosophila homeotic genes structurally related to the yeast transcriptional activator SNF2SWI2

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