Affiliation:
1. School of Chemistry South China Normal University GDMPA Key Laboratory for Process Control and Quality Evaluation of Chiral Pharmaceuticals Guangzhou Key Laboratory of Analytical Chemistry for Biomedicine Key Laboratory of Theoretical Chemistry of Environment Ministry of Education Guangzhou Guangdong 510006 P. R. China
Abstract
AbstractHydroiodic acid‐mediated vicinal iodosulfonylation reaction of alkynes with sodium sulfinates is proposed for the synthesis of (E)‐β‐iodovinyl sulfones. The method is easy to operate, environmentally friendly, using inexpensive and easily available raw materials, and giving the target products with good regio‐ and stereoselectivity in satisfactory yields.
Funder
Basic and Applied Basic Research Foundation of Guangdong Province
National Natural Science Foundation of China