Quantitation of unbound sunitinib and its metaboliteN-desethyl sunitinib (SU12662) in human plasma by equilibrium dialysis and liquid chromatography-tandem mass spectrometry: application to a pharmacokinetic study

Author:

Rais Rana1,Zhao Ming1,He Ping1,Xu Linping1,Deeken John F.2,Rudek Michelle A.1

Affiliation:

1. The Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins; Baltimore; MD; 21231; USA

2. Lombardi Cancer Center; Georgetown University Medical Center; Washington; DC; 20007; USA

Publisher

Wiley

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,General Medicine,Biochemistry,Analytical Chemistry

Reference21 articles.

1. Role of tyrosine kinase inhibitors in cancer therapy;Arora;Journal of Pharmacology and Experimental Therapeutics,2005

2. Sunitinib malate for the treatment of metastatic renal cell carcinoma and gastrointestinal stromal tumors;Adams;Clinical Therapeutics,2007

3. Sunitinib maleate;Atkins;Nature Review Drug Discovery,2006

4. Equilibrium dialysis, ultrafiltration, and ultracentrifugation compared for determining the plasma-protein-binding characteristics of valproic acid;Barre;Clinical Chemistry,1985

5. Measurement of fraction unbound paclitaxel in human plasma;Brouwer;Drug Metabolism and Disposition,2000

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