Structure-Activity Relationship Studies of CNS Agents, Part 26 4-[2-(Cycloalkanecarboxamido)ethyl]-1-(2-methoxyphenyl)-piperazines: High-Affinity 5-HT1A Agonists-Reference-Cited by-同舟云学术

Structure-Activity Relationship Studies of CNS Agents, Part 26 4-[2-(Cycloalkanecarboxamido)ethyl]-1-(2-methoxyphenyl)-piperazines: High-Affinity 5-HT1A Agonists

Published:1995 Issue:11-12 Volume:328 Page:770-774
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:de
Short-container-title:Arch. Pharm. Pharm. Med. Chem.

Author:

Mokrosz Jerzy L.,Paluchowska Maria H.,Klodzińska Aleksandra,Charakchieva-Minol Sijka,Chojnacka-Wójcik Ewa

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Reference23 articles.

1. Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands

2. N-(phthalimidoalkyl) derivatives of serotonergic agents: a common interaction at 5-HT1A serotonin binding sites?

3. The behavioural, but not the hypothermic or corticosterone, response to 8-hydroxy-2-(di-n-propylamino)-tetralin, is antagonized by nan-190 in the rat

4. The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro

5. Concepts for the design of 5-HT1A serotonin agonists and antagonists

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