Phenotypic Identification of a Novel Autophagy Inhibitor Chemotype Targeting Lipid Kinase VPS34

Author:

Robke Lucas12,Laraia Luca1,Carnero Corrales Marjorie A.12,Konstantinidis Georgios3,Muroi Makoto45,Richters André2,Winzker Michael12,Engbring Tobias2,Tomassi Stefano2,Watanabe Nobumoto56,Osada Hiroyuki45,Rauh Daniel2,Waldmann Herbert12ORCID,Wu Yao-Wen3,Engel Julian2

Affiliation:

1. Max-Planck-Institute of Molecular Physiology; Department of Chemical Biology; Otto-Hahn-Strasse 11 44227 Dortmund Germany

2. Faculty of Chemistry and Chemical Biology; TU Dortmund University; Otto-Hahn-Strasse 4a 44227 Dortmund Germany

3. Chemical Genomics Centre of the Max-Planck-Society; Otto-Hahn-Strasse 15 44227 Dortmund Germany

4. Chemical Biology Research Group; RIKEN CSRS; 2-1, Hirosawa, Wako Saitama 351-0198 Japan

5. RIKEN-Max Planck Joint Research Division for Systems Chemical Biology; RIKEN CSRS; 2-1, Hirosawa, Wako Saitama 351-0198 Japan

6. Bio-Active Compounds Discovery Research Unit; RIKEN CSRS; 2-1, Hirosawa, Wako Saitama 351-0198 Japan

Funder

Boehringer Ingelheim Fonds (DE)

Alexander von Humboldt-Stiftung

Schweizerischer Nationalfonds zur Förderung der Wissenschaftlichen Forschung

Fonds der Chemischen Industrie

European Research Council (ChemBioAP)

Behrens-Weise-Stiftung

Publisher

Wiley

Subject

General Chemistry,Catalysis

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