Quantitative Prediction of Rate Constants for Aqueous Racemization To Avoid Pointless Stereoselective Syntheses-Reference-Cited by-同舟云学术

Quantitative Prediction of Rate Constants for Aqueous Racemization To Avoid Pointless Stereoselective Syntheses

Published:2017-11-15 Issue:4 Volume:57 Page:982-985
ISSN:1433-7851
Container-title:Angewandte Chemie International Edition
language:en
Short-container-title:Angew. Chem. Int. Ed.

Author:

Ballard Andrew¹,Ahmad Hiwa O.¹²,Narduolo Stefania¹,Rosa Lucy³,Chand Nikki³,Cosgrove David A.³,Varkonyi Peter⁴,Asaad Nabil³,Tomasi Simone⁵,Buurma Niklaas J.¹,Leach Andrew G.⁶^ORCID

Affiliation:

1. Physical Organic Chemistry Centre; School of Chemistry; Cardiff University; Main Building, Park Place, Cardiff CF10 3AT UK

2. Pharmaceutical Chemistry Department; College of Pharmacy; Hawler Medical University; Erbil Kurdistan Region Iraq

3. AstraZeneca Pharmaceuticals, Mereside; Alderley Park Macclesfield SK10 4TG UK

4. AstraZeneca R+D; Pepparedsleden 1 43183 Mölndal Sweden

5. AstraZeneca; Charter Way, Silk Road Business Park Macclesfield SK10 2NA UK

6. School of Pharmacy and Biomolecular Sciences; Liverpool John Moores University; Liverpool L3 3AF UK

Funder

Engineering and Physical Sciences Research Council (EPSRC)

Publisher

Wiley

Subject

General Chemistry,Catalysis

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/anie.201709163/fullpdf

Reference36 articles.

1. Chiral Inversion and Hydrolysis of Thalidomide: Mechanisms and Catalysis by Bases and Serum Albumin, and Chiral Stability of Teratogenic Metabolites

2. Dynamic Kinetic Resolution (DKR)

3. Dynamic kinetic resolution

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