Small-Molecule-Mediated Degradation of the Androgen Receptor through Hydrophobic Tagging-Reference-Cited by-同舟云学术

Small-Molecule-Mediated Degradation of the Androgen Receptor through Hydrophobic Tagging

Published:2015-06-17 Issue:33 Volume:54 Page:9659-9662
ISSN:1433-7851
Container-title:Angewandte Chemie International Edition
language:en
Short-container-title:Angew. Chem. Int. Ed.

Author:

Gustafson Jeffrey L.,Neklesa Taavi K.,Cox Carly S.,Roth Anke G.,Buckley Dennis L.,Tae Hyun Seop,Sundberg Thomas B.,Stagg D. Blake,Hines John,McDonnell Donald P.,Norris John D.,Crews Craig M.

Publisher

Wiley

Subject

General Chemistry,Catalysis

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/anie.201503720/fullpdf

Reference33 articles.

1. A Dual Small-Molecule Rheostat for Precise Control of Protein Concentration in Mammalian Cells

2. Targeting the Undruggable Proteome: The Small Molecules of My Dreams

3. Overcoming mutation-based resistance to antiandrogens with rational drug design

4. Strategies for silencing human disease using RNA interference

5. Current prospects for RNA interference-based therapies

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