Bioactive Macrocyclic Inhibitors of the PD-1/PD-L1 Immune Checkpoint

Author:

Magiera-Mularz Katarzyna1,Skalniak Lukasz1,Zak Krzysztof M.23,Musielak Bogdan1,Rudzinska-Szostak Ewa4,Berlicki Łukasz4,Kocik Justyna1,Grudnik Przemyslaw23,Sala Dominik1,Zarganes-Tzitzikas Tryfon5,Shaabani Shabnam5,Dömling Alexander5,Dubin Grzegorz23,Holak Tad A.16

Affiliation:

1. Department of Organic Chemistry; Faculty of Chemistry; Jagiellonian University; Ingardena 3 30-060 Krakow Poland

2. Malopolska Centre of Biotechnology; Jagiellonian University; Gronostajowa 7a 30-387 Krakow Poland

3. Faculty of Biochemistry, Biophysics and Biotechnology; Jagiellonian University; Gronostajowa 7 30-387 Krakow Poland

4. Department of Bioorganic Chemistry; Faculty of Chemistry; Wrocław University of Science and Technology; Wybrzeże Wyspiańskiego 27 50-370 Wrocław Poland

5. Department for Drug Design; University of Groningen; A. Deusinglaan 9 AV 9713 Groningen The Netherlands

6. Max Planck Institute for Biochemistry; Am Klopferspitz 18a 82152 Martinsried Germany

Funder

Narodowe Centrum Nauki

European Community Framework Programme

National Institutes of Health

Co-funding of regional, national and international programmes (COFUND)

European Union structural funds

European Regional Development Fund

Publisher

Wiley

Subject

General Chemistry,Catalysis

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