Mechanism-Based Inhibitors of the Human Sirtuin 5 Deacylase: Structure-Activity Relationship, Biostructural, and Kinetic Insight-Reference-Cited by-同舟云学术

Mechanism-Based Inhibitors of the Human Sirtuin 5 Deacylase: Structure-Activity Relationship, Biostructural, and Kinetic Insight

Published:2017-11-02 Issue:47 Volume:56 Page:14836-14841
ISSN:1433-7851
Container-title:Angewandte Chemie International Edition
language:en
Short-container-title:Angew. Chem. Int. Ed.

Author:

Rajabi Nima¹^ORCID,Auth Marina¹,Troelsen Kathrin R.¹,Pannek Martin²,Bhatt Dhaval P.³,Fontenas Martin¹,Hirschey Matthew D.³,Steegborn Clemens²,Madsen Andreas S.¹^ORCID,Olsen Christian A.¹^ORCID

Affiliation:

1. Center for Biopharmaceuticals & Department of Drug Design and Pharmacology; University of Copenhagen; Universitetsparken 2 2100 Copenhagen Denmark

2. Universität Bayreuth; Lehrstuhl Biochemie und Forschungszentrum für Biomakromoleküle; Universitätsstrasse 30 95447 Bayreuth Germany

3. Duke University Medical Center; Sarah W. Stedman Nutrition and Metabolism Center; 4321 Medical Park Drive Durham NC 27704 USA

Funder

Carlsbergfondet

Lundbeckfonden

Novo Nordisk Fonden (DK)

H2020 European Research Council

Oberfrankenstiftung

Publisher

Wiley

Subject

General Chemistry,Catalysis

Reference51 articles.

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