In silicoprediction of drug dissolution and absorption with variation in intestinal pH for BCS class II weak acid drugs: ibuprofen and ketoprofen-Reference-Cited by-同舟云学术

In silicoprediction of drug dissolution and absorption with variation in intestinal pH for BCS class II weak acid drugs: ibuprofen and ketoprofen

Published:2012-08-21 Issue:7 Volume:33 Page:366-377
ISSN:0142-2782
Container-title:Biopharmaceutics & Drug Disposition
language:en
Short-container-title:Biopharm. Drug Dispos.

Author:

Tsume Yasuhiro¹,Langguth Peter²,Garcia-Arieta Alfredo³,Amidon Gordon L.¹

Affiliation:

1. College of Pharmacy; University of Michigan; Ann Arbor; Michigan; 48109-1065; USA

2. Department of Pharmaceutical Technology and Biopharmaceutics; Johannes Gutenberg-University of Mainz; Staudinger Weg 5; Mainz; D-55099; Germany

3. Division de Farmacologia y Evaluacion Clinica, Subdireccion General de Medicamentos de Uso Humano; Agencia Espanola de Medicamentos y Productos Sanitarios; C/ Campezo 1, Edifico 8; 28022; Madrid; Spain

Publisher

Wiley

Subject

Pharmacology (medical),Pharmaceutical Science,Pharmacology,General Medicine

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/bdd.1800/fullpdf

Reference50 articles.

1. U.S. FDA Department of Health and Human Services Food and Drug Administration Center for Evaluation and Research Guidances for Industry: Waiver of In Vivo Bioavailability and Bioequivalence Studies for Immediate-release Solid Oral Dosage Forms Based on a Biopharmaceutics Classification System 2000

2. EMA Guideline on the Investigation of Bioequivalence 2010

3. A theoretical basis for a biopharmaceutic drug classification: the correlation of in vitro drug product dissolution and in vivo bioavailability;Amidon;Pharm Res,1995

4. The ‘high solubility’ definition of the current FDA Guidance on Biopharmaceutical Classification System may be too strict for acidic drugs;Yazdanian;Pharm Res,2004

5. Review of global regulations concerning biowaivers for immediate release solid oral dosage forms;Gupta;Eur J Pharm Sci,2006

Cited by 86 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A Fast HPLC/UV Method for Determination of Ketoprofen in Cellular Media.;ChemistryOpen;2023-11-13

2. Use of In silico Methodologies to Predict the Bioavailability of Oral Suspensions: A Regulatory Approach;Current Pharmaceutical Design;2023-10

3. How bio-relevant buffering media affect dissolution and release kinetics of solid formula: Ibuprofen as a model;Journal of Drug Delivery Science and Technology;2023-09

4. The influence of formulation and hardness on the dissolution rate of ketoprofen in prolonged release tablets;Macedonian Pharmaceutical Bulletin;2023-09

5. Predictive Potential of Acido-Basic Properties, Solubility and Food on Bioequivalence Study Outcome: Analysis of 128 Studies;Drugs in R&D;2023-06-10