Drofenine: a 2‐APB analog with improved selectivity for human TRPV3-Reference-Cited by-同舟云学术

Drofenine: a 2‐APB analog with improved selectivity for human TRPV3

Published:2014-07-02 Issue:5 Volume:2 Page:
ISSN:2052-1707
Container-title:Pharmacology Research & Perspectives
language:en
Short-container-title:Pharmacol Res Perspect

Author:

Deering‐Rice Cassandra E.¹,Mitchell Virginia K.¹,Romero Erin G.¹,Abdel Aziz May H.¹,Ryskamp Daniel A.²,Križaj David²,Venkat Raj Gopal³,Reilly Christopher A.¹

Affiliation:

1. Department of Pharmacology and Toxicology University of Utah Salt Lake City Utah 84112

2. Department of Ophthalmology and Visual Sciences Interdepartmental Neuroscience Program University of Utah Salt Lake City Utah 84132

3. Department of Medicinal Chemistry University of Utah Salt Lake City Utah 84112

Funder

National Institute of Environmental Health Sciences

Publisher

Wiley

Subject

General Pharmacology, Toxicology and Pharmaceutics,Neurology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/prp2.62

Reference35 articles.

1. The Mechanosensitive Ion Channel Piezo1 Is Inhibited by the Peptide GsMTx4

2. Farnesyl Pyrophosphate Is a Novel Pain-producing Molecule via Specific Activation of TRPV3

3. Isopentenyl pyrophosphate is a novel antinociceptive substance that inhibits TRPV3 and TRPA1 ion channels

4. 17(R)-resolvin D1 specifically inhibits transient receptor potential ion channel vanilloid 3 leading to peripheral antinociception

5. 2‐Aminoethoxydiphenyl borate (2‐APB) is a reliable blocker of store‐operated Ca2+entry but an inconsistent inhibitor of InsP3‐induced Ca2+release

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