Analysis of full and partial agonists binding to β2-adrenergic receptor suggests a role of transmembrane helix V in agonist-specific conformational changes-Reference-Cited by-同舟云学术

Analysis of full and partial agonists binding to β2-adrenergic receptor suggests a role of transmembrane helix V in agonist-specific conformational changes

Published:2009-04-07 Issue:4 Volume:22 Page:307-318
ISSN:0952-3499
Container-title:Journal of Molecular Recognition
language:en
Short-container-title:J. Mol. Recognit.

Author:

Katritch Vsevolod,Reynolds Kimberly A.,Cherezov Vadim,Hanson Michael A.,Roth Christopher B.,Yeager Mark,Abagyan Ruben

Publisher

Wiley

Subject

Molecular Biology,Structural Biology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/jmr.949/fullpdf

Reference50 articles.

1. Biased probability Monte Carlo conformational searches and electrostatic calculations for peptides and proteins;Abagyan;J. Mol. Biol.,1994

2. Icm: a new method for protein modeling and design: applications to docking and structure prediction from the distorted native conformation;Abagyan;J. Comp. Chem.,1994

3. Catechol-binding serines of beta(2)-adrenergic receptors control the equilibrium between active and inactive receptor states;Ambrosio;Mol. Pharmacol.,2000

4. The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors;Baker;Br. J. Pharmacol.,2005

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