Synthesis of C-14 labeled GABAAα2/α3 selective partial agonists and the investigation of late-occurring and long-circulating metabolites of GABAAreceptor modulator AZD7325-Reference-Cited by-同舟云学术

Synthesis of C-14 labeled GABAAα2/α3 selective partial agonists and the investigation of late-occurring and long-circulating metabolites of GABAAreceptor modulator AZD7325

Published:2018-03-30 Issue:5 Volume:61 Page:415-426
ISSN:0362-4803
Container-title:Journal of Labelled Compounds and Radiopharmaceuticals
language:en
Short-container-title:J Label Compd Radiopharm

Author:

Artelsmair Markus¹^ORCID,Gu Chungang²,Lewis Richard J.³^ORCID,Elmore Charles S.¹^ORCID

Affiliation:

1. Early Chemical Development, Pharmaceutical Sciences, IMED Biotech Unit; AstraZeneca; Gothenburg Sweden

2. DMPK, Oncology, IMED Biotech Unit; AstraZeneca; Boston MA USA

3. Medicinal Chemistry, Respiratory, Inflammation and Autoimmunity, IMED Biotech Unit; AstraZeneca; Gothenburg Sweden

Funder

H2020 Marie Skłodowska-Curie Actions

Marie Sklodowska-Curie

Publisher

Wiley

Subject

Organic Chemistry,Spectroscopy,Drug Discovery,Radiology Nuclear Medicine and imaging,Biochemistry,Analytical Chemistry

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