Synthesis and Biological Evaluation of Tripartin, a Putative KDM4 Natural Product Inhibitor, and 1-Dichloromethylinden-1-ol Analogues-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of Tripartin, a Putative KDM4 Natural Product Inhibitor, and 1-Dichloromethylinden-1-ol Analogues

Published:2018-08-21 Issue:18 Volume:13 Page:1949-1956
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Guillade Lucía¹,Sarno Federica²,Tarhonskaya Hanna³,Nebbioso Angela²,Alvarez Susana¹,Kawamura Akane³,Schofield Christopher J.³,Altucci Lucia²,de Lera Ángel R.¹^ORCID

Affiliation:

1. Departamento de Química Orgánica, Facultade de Química, CINBIO and IBIV; Universidade de Vigo; Campus As Lagoas-Marcosende 36310 Vigo Spain

2. Università degli Studi della Campania “Luigi Vanvitelli”; Vico L. De Crecchio 7 80138 Napoli Italy

3. Chemistry Research Laboratory, Department of Chemistry; University of Oxford; Mansfield Road Oxford OX1 3TA UK

Funder

Ministerio de Economía y Competitividad

MIUR-Italian Ministry of Education

Associazione Italiana per la Ricerca sul Cancro

Erzincan Üniversitesi

Cancer Research UK

Wellcome Trust

Consellería de Cultura, Educación e Ordenación Universitaria, Xunta de Galicia

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201800377/fullpdf

Reference67 articles.

1. Histone Lysine Methylation Dynamics: Establishment, Regulation, and Biological Impact

2. Targeting histone methyltransferases and demethylases in clinical trials for cancer therapy

3. Selective Inhibitors of Protein Methyltransferases

Cited by 13 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Total Synthesis, structure revision and antifungal activity of palmarumycin B8 and B7;Bioorganic Chemistry;2024-07

2. Total Synthesis and Biological Activity of (±)-Guignardin A, (±)-Palmarumycin B₉, and Their Derivatives;ACS Agricultural Science & Technology;2024-02-27

3. A Diastereoselective Assembly of Tetralone Derivatives via a Tandem Michael Reaction and ipso-Substitution of the Nitro Group;The Journal of Organic Chemistry;2023-04-17

4. Inhibitors of Jumonji-C domain-containing histone demethylases;Epigenetic Cancer Therapy;2023

5. Recent Advances with KDM4 Inhibitors and Potential Applications;Journal of Medicinal Chemistry;2022-07-15