Bicyclic Derivatives of the Potent Dual Aromatase-Steroid Sulfatase Inhibitor 2-Bromo-4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities-Reference-Cited by-同舟云学术

Bicyclic Derivatives of the Potent Dual Aromatase-Steroid Sulfatase Inhibitor 2-Bromo-4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities

Published:2010-07-14 Issue:9 Volume:5 Page:1577-1593
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Wood Paul M.,Woo L. W. Lawrence,Labrosse Jean-Robert,Thomas Mark P.,Mahon Mary F.,Chander Surinder K.,Purohit Atul,Reed Michael J.,Potter Barry V. L.

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201000203/fullpdf

Reference55 articles.

1. ON THE TREATMENT OF INOPERABLE CASES OF CARCINOMA OF THE MAMMA: SUGGESTIONS FOR A NEW METHOD OF TREATMENT, WITH ILLUSTRATIVE CASES.1

2. Aromatase inhibitors in breast cancer

3. Nonsteroidal aromatase inhibitors: Recent advances

4. Aromatase Inhibitors in the Treatment of Breast Cancer

5. Aromatase inhibitors in early breast cancer therapy: a variety of treatment strategies

Cited by 27 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Secosteroid thiosemicarbazides and secosteroid–1,2,4-triazoles as antiproliferative agents targeting breast cancer cells: Synthesis and biological evaluation;The Journal of Steroid Biochemistry and Molecular Biology;2023-11

2. Dual aromatase-steroid sulfatase inhibitors (DASI's) for the treatment of breast cancer: a structure guided ligand based designing approach;Journal of Biomolecular Structure and Dynamics;2022-12-12

3. Dual Targeting of Steroid Sulfatase and 17β-Hydroxysteroid Dehydrogenase Type 1 by a Novel Drug-Prodrug Approach: A Potential Therapeutic Option for the Treatment of Endometriosis;Journal of Medicinal Chemistry;2022-08-22

4. Dual Aromatase-Sulphatase Inhibitors (DASIs) for the Treatment of Hormone Dependent Breast Cancer;Mini-Reviews in Medicinal Chemistry;2021-12

5. Steroid Sulphatase and Its Inhibitors: Past, Present and Future;Molecules;2021-05-11