Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist-Reference-Cited by-同舟云学术

Discovery of 1-(2,4-Dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a Potential Peripheral Cannabinoid-1 Receptor Inverse Agonist

Published:2010-07-22 Issue:9 Volume:5 Page:1439-1443
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Hung Ming-Shiu,Chang Chun-Ping,Li Ting-Chieh,Yeh Teng-Kuang,Song Jen-Shin,Lin Yinchiu,Wu Chien-Huang,Kuo Po-Chu,Amancha Prashanth K.,Wong Ying-Chieh,Hsiao Wen-Chi,Chao Yu-Sheng,Shia Kak-Shan

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201000246/fullpdf

Reference28 articles.

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4. Molecular characterization of a peripheral receptor for cannabinoids

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