Discovery and Pharmacophore Mapping of a Low‐Nanomolar Inhibitor of P. falciparum Growth-Reference-Cited by-同舟云学术

Discovery and Pharmacophore Mapping of a Low‐Nanomolar Inhibitor of P. falciparum Growth

Published:2019-11-12 Issue:23 Volume:14 Page:1982-1994
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Bassanini Ivan¹²^ORCID,Parapini Silvia³²^ORCID,Galli Corinna¹²,Vaiana Nadia¹²,Pancotti Andrea¹²,Basilico Nicoletta³²^ORCID,Taramelli Donatella⁴²^ORCID,Romeo Sergio¹²^ORCID

Affiliation:

1. Dipartimento di Scienze FarmaceuticheUniversità degli Studi di Milano Via Mangiagalli 25 20133 Milan Italy

2. Centro Interuniversitario di Ricerca sulla Malaria-Italian Malaria Network

3. Dipartimento di Scienze Biomediche, Chirurgiche e OdontoiatricheUniversità degli Studi di Milano Via Pascal, 36 20133 Milan Italy

4. Dipartimento di Scienze Farmacologiche e BiomolecolariUniversità degli Studi di Milano Via Pascal 36 20133 Milan Italy

Funder

Università degli Studi di Milano

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201900526

Reference20 articles.

1. Innate sensing of malaria parasites

2. World Health Organization WORLD MALARIA REPORT 2018 n.d.

3. Multiple populations of artemisinin-resistant Plasmodium falciparum in Cambodia

4. Antimalarial Drug Resistance: Literature Review and Activities and Findings of the ICEMR Network

5. High Antiplasmodial Activity of Novel Plasmepsins I and II Inhibitors

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