Synthesis, Biochemistry, and Computational Studies of Brominated Thienyl Chalcones: A New Class of Reversible MAO-B Inhibitors-Reference-Cited by-同舟云学术

Synthesis, Biochemistry, and Computational Studies of Brominated Thienyl Chalcones: A New Class of Reversible MAO-B Inhibitors

Published:2016-05-09 Issue:11 Volume:11 Page:1161-1171
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Mathew Bijo¹^ORCID,Haridas Abitha²,Uçar Gülberk³,Baysal Ipek³,Joy Monu⁴,Mathew Githa E.⁵,Lakshmanan Baskar²,Jayaprakash Venkatesan⁶

Affiliation:

1. Division of Drug Design and Medicinal Chemistry Research Laboratory; Department of Pharmaceutical Chemistry; Ahalia School of Pharmacy; Palakkad 678557 Kerala India

2. Department of Pharmaceutical Chemistry; Grace College of Pharmacy; Palakkad 678004 Kerala India

3. Department of Biochemistry; Faculty of Pharmacy; Hacettepe University; 06100 Sıhhiye Ankara Turkey

4. School of Pure & Applied Physics; Mahatma Gandhi University; Kottayam 686560 India

5. Department of Pharmacology; Grace College of Pharmacy; Palakkad 678004 Kerala India

6. Department of Pharmaceutical Sciences and Technology; Birla Institute of Technology; Mesra, Ranchi 835215 Jharkhand India

Funder

Institute for Intensive Research in Basic Sciences (IIRBS), Mahatma Gandhi University

Sophisticated Analytical Instrument Facility, Indian Institute of Technology

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Reference52 articles.

1. Enzymology of monoamine oxidase

2. 8-Substituted 3-Arylcoumarins as Potent and Selective MAO-B Inhibitors: Synthesis, Pharmacological Evaluation, and Docking Studies

3. Proposed structural basis of interaction of piperine and related compounds with monoamine oxidases

4. MONOAMINE OXIDASE: From Genes to Behavior

5. Drug treatment of Parkinson’s disease

Cited by 75 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Dual-target inhibitors based on acetylcholinesterase: Novel agents for Alzheimer's disease;European Journal of Medicinal Chemistry;2024-12

2. Chalcones with N‐Methylpiperazine Moiety: Synthesis, Monoamine Oxidase Inhibition, Neuroprotective Effect and Computer Simulation Study;ChemistrySelect;2024-04-09

3. Probing the inhibition of MAO-B by chalcones: an integrated approach combining molecular docking, ADME analysis, MD simulation, and MM-PBSA calculations;Journal of Molecular Modeling;2024-03-13

4. Redefining Chalcone Synthesis: Aldol Adduct Elimination for the Rapid Access to Thienyl Chalcones;ACS Omega;2024-03-12

5. Development of morpholine ring-bearing halogenated α,β-unsaturated ketones as selective monoamine oxidase-B inhibitors;Applied Biological Chemistry;2024-01-22