Discovery of 5′′-Chloro-N-[(5,6-dimethoxypyridin-2-yl)methyl]-2,2′:5′,3′′-terpyridine-3′-carboxamide (MK-1064): A Selective Orexin 2 Receptor Antagonist (2-SORA) for the Treatment of Insomnia-Reference-Cited by-同舟云学术

Discovery of 5′′-Chloro-N-[(5,6-dimethoxypyridin-2-yl)methyl]-2,2′:5′,3′′-terpyridine-3′-carboxamide (MK-1064): A Selective Orexin 2 Receptor Antagonist (2-SORA) for the Treatment of Insomnia

Published:2013-12-27 Issue:2 Volume:9 Page:311-322
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Roecker Anthony J.,Mercer Swati P.,Schreier John D.,Cox Christopher D.,Fraley Mark E.,Steen Justin T.,Lemaire Wei,Bruno Joseph G.,Harrell C. Meacham,Garson Susan L.,Gotter Anthony L.,Fox Steven V.,Stevens Joanne,Tannenbaum Pamela L.,Prueksaritanont Thomayant,Cabalu Tamara D.,Cui Donghui,Stellabott Joyce,Hartman George D.,Young Steven D.,Winrow Christopher J.,Renger John J.,Coleman Paul J.

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201300447/fullpdf

Reference93 articles.

1. Diagnosis and treatment of insomnia

2. Conductas complejas durante el sueño inducidas por zolpidem

3. Overview of Experimental and Conventional Pharmacological Approaches in the Treatment of Sleep and Wake Disorders

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