Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1H )-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions-Reference-Cited by-同舟云学术

Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1H )-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions

Published:2018-09-17 Issue:20 Volume:13 Page:2217-2228
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Pedron Julien¹,Boudot Clotilde²,Bourgeade-Delmas Sandra³,Sournia-Saquet Alix¹,Paloque Lucie¹,Rastegari Maryam¹,Abdoulaye Mansour¹,El-Kashef Hussein⁴,Bonduelle Colin¹,Pratviel Geneviève¹,Wyllie Susan⁵,Fairlamb Alan H.⁵,Courtioux Bertrand²,Verhaeghe Pierre¹^ORCID,Valentin Alexis³

Affiliation:

1. LCC-CNRS; Université de Toulouse, CNRS; UPS; 205 route de Narbonne 31077 Toulouse France

2. Université de Limoges; UMR INSERM 1094; Neuroépidémiologie Tropicale; Faculté de Pharmacie; 2 rue du Dr Marcland 87025 Limoges France

3. UMR 152 PharmaDev; Université de Toulouse, IRD; UPS; 35 Chemin des Maraîchers 31400 Toulouse France

4. Assiut University; Faculty of Science; Department of Chemistry; 71516 Assiut Egypt

5. University of Dundee; School of Life Sciences; Division of Biological Chemistry and Drug Discovery; Dow Street Dundee DD1 5EH UK

Funder

Wellcome Trust

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201800456/fullpdf

Reference40 articles.

1. Differences between Trypanosoma brucei gambiense Groups 1 and 2 in Their Resistance to Killing by Trypanolytic Factor 1

2. Human African trypanosomiasis

3. Leishmaniasis

4. Visceral leishmanisis in paediatrics: a study of 367 cases in southwest Iran

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis, molecular docking analysis and in-vitro evaluation of 1,4-dihydroxyanthraquinone derivatives as anti-trypanosomal agents;Letters in Organic Chemistry;2022-11-14

2. The Potential of 2-Substituted Quinolines as Antileishmanial Drug Candidates;Molecules;2022-04-02

3. Unveiling the relevance of the redox character of nitroaromatic and nitroheteroaromatic compounds as potential medicines;Current Opinion in Electrochemistry;2021-10

4. Synthesis, Structure and In Vitro Anti-Trypanosomal Activity of Non-Toxic Arylpyrrole-Based Chalcone Derivatives;Molecules;2020-04-04

5. New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi;ACS Medicinal Chemistry Letters;2020-02-06