NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family-Reference-Cited by-同舟云学术

NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family

Published:2018-07-20 Issue:16 Volume:13 Page:1629-1633
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Tröster Alix¹,Heinzlmeir Stephanie²³,Berger Benedict-Tilman⁴⁵^ORCID,Gande Santosh L.¹³,Saxena Krishna¹,Sreeramulu Sridhar¹,Linhard Verena¹,Nasiri Amir H.¹,Bolte Michael⁶^ORCID,Müller Susanne⁴,Kuster Bernhard²³,Médard Guillaume²^ORCID,Kudlinzki Denis¹³,Schwalbe Harald¹³^ORCID

Affiliation:

1. Center for Biomolecular Magnetic Resonance (BMRZ); Institute for Organic Chemistry and Chemical Biology; Johann Wolfgang Goethe University; Max-von-Laue-Straße 7 60438 Frankfurt am Main Germany

2. Chair of Proteomics and Bioanalytics; Technical University of Munich; Emil-Erlenmeyer-Forum 5 85354 Freising Germany

3. German Cancer Consortium (DKTK); German Cancer Research Center (DKFZ); Im Neuenheimer Feld 280 69120 Heidelberg Germany

4. Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences; Goethe University Frankfurt; Frankfurt am Main Germany

5. Institute for Pharmaceutical Chemistry; Johann Wolfgang Goethe University; Max-von-Laue-Straße 9 60438 Frankfurt am Main Germany

6. Institute for Inorganic Chemistry; Goethe University Frankfurt; Frankfurt am Main Germany

Funder

Structural Genomics Consortium

German consortium for translational cancer research (DKTK)

DFG (SFB807)

EU research infrastructure iNEXT

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201800398/fullpdf

Reference36 articles.

1. Ectodomain structures of Eph receptors

2. Eph/ephrin molecules—a hub for signaling and endocytosis

3. Eph receptors and ephrins in cancer: bidirectional signalling and beyond

4. Eph Receptors and Ephrins: Therapeutic Opportunities

5. Eph Receptors and Ephrins in Cancer: Common Themes and Controversies

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