Structure‐Based Screening of Tetrazolylhydrazide Inhibitors versus KDM4 Histone Demethylases-Reference-Cited by-同舟云学术

Structure‐Based Screening of Tetrazolylhydrazide Inhibitors versus KDM4 Histone Demethylases

Published:2019-10-10 Issue:21 Volume:14 Page:1828-1839
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Małecki Piotr H.¹²³^ORCID,Rüger Nicole⁴,Roatsch Martin⁵⁶^ORCID,Krylova Oxana⁷,Link Andreas⁴^ORCID,Jung Manfred⁵^ORCID,Heinemann Udo²^ORCID,Weiss Manfred S.¹^ORCID

Affiliation:

1. Macromolecular Crystallography Helmholtz-Zentrum Berlin für Materialien und Energie Albert-Einstein-Str. 15 12489 Berlin Germany

2. Macromolecular Structure and Interaction Max Delbrück Center for Molecular Medicine Robert-Rössle-Str. 10 13125 Berlin Germany

3. Current address: International Institute of Molecular and Cell Biology Ks. Trojdena Street 4 02-109 Warsaw Poland

4. Institute of Pharmacy Universität Greifswald Friedrich-Ludwig-Jahn-Str. 17 17489 Greifswald Germany

5. Institute of Pharmaceutical Sciences University of Freiburg Albertstr. 25 79104 Freiburg Germany

6. Current address: Københavns Universitet Center for Biopharmaceuticals Universitetsparken 2 2100 Copenhagen Denmark

7. Department of Molecular Biophysics Forschungsinstitut für Molekulare Pharmakologie Robert-Rössle-Str. 10 13125 Berlin Germany

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201900441

Reference74 articles.

1. The genetic control of wing development inDrosophila

3. Epigenetic protein families: a new frontier for drug discovery

4. Epigenetic control of the immune system: histone demethylation as a target for drug discovery

5. Chromatin targeting drugs in cancer and immunity

Cited by 15 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structure-based mapping of the histone-binding pocket of KDM4D using functionalized tetrazole and pyridine core compounds;European Journal of Medicinal Chemistry;2024-10

2. Innovative synthesis of drug-like molecules using tetrazole as core building blocks;Beilstein Journal of Organic Chemistry;2024-04-29

3. Microwave Assisted Synthesis, Spectro-Analytical, Docking and Anti Microbial Studies of Tetrazole Linked N-Acyl Hydrazone Derivatives;2024

4. Synthesis, characterization, DNA binding, protein binding, antioxidant and anti microbial activity of tetrazole ring based complexes;Journal of Molecular Structure;2023-11

5. Development of JmjC-domain-containing histone demethylase (KDM2-7) inhibitors for cancer therapy;Drug Discovery Today;2023-05