[Carboxyl -11 C]Labelling of Four High-Affinity cPLA2α Inhibitors and Their Evaluation as Radioligands in Mice by Positron Emission Tomography-Reference-Cited by-同舟云学术

[Carboxyl -11 C]Labelling of Four High-Affinity cPLA2α Inhibitors and Their Evaluation as Radioligands in Mice by Positron Emission Tomography

Published:2018-01-10 Issue:2 Volume:13 Page:138-146
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Fisher Martin J.¹,McMurray Lindsay¹,Lu Shuiyu²^ORCID,Morse Cheryl L.²,Liow Jeih-San²,Zoghbi Sami S.²,Kowalski Aneta²,Tye George L.²,Innis Robert B.²,Aigbirhio Franklin I.¹,Pike Victor W.²^ORCID

Affiliation:

1. Molecular Imaging Chemistry Laboratory, Wolfson Brain Imaging Centre; University of Cambridge; Cambridge Biomedical Campus Cambridge CB2 0QQ UK

2. Molecular Imaging Branch; National Institute of Mental Health, National Institutes of Health; 10 Center Drive, Room B3C346 Bethesda MD 20892 USA

Funder

National Institutes of Health

Medical Research Council

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201700697/fullpdf

Reference62 articles.

1. Cytosolic phospholipase A2

2. Cytosolic phospholipase A2: physiological function and role in disease

3. Phospholipase A2 Enzymes: Physical Structure, Biological Function, Disease Implication, Chemical Inhibition, and Therapeutic Intervention

4. Inhibitors of Brain Phospholipase A2Activity: Their Neuropharmacological Effects and Therapeutic Importance for the Treatment of Neurologic Disorders

5. Cytosolic phospholipase A2 as a mediator of disease pathogenesis

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The development of 11C-carbonylation chemistry: A systematic view;Nuclear Medicine and Biology;2021-01

2. A General and Scalable Synthesis of Polysubstituted Indoles;Molecules;2020-11-28

3. Copper(I)-Mediated 11C-Carboxylation of (Hetero)arylstannanes;ACS Omega;2020-04-02

4. [11C]Carbon monoxide: advances in production and application to PET radiotracer development over the past 15 years;EJNMMI Radiopharmacy and Chemistry;2019-09-18

5. Small-molecule inhibitors as potential therapeutics and as tools to understand the role of phospholipases A2;Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids;2019-06