Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase-Reference-Cited by-同舟云学术

Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase

Published:2017-04-12 Issue:16 Volume:12 Page:1359-1368
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Madia Valentina Noemi¹^ORCID,Benedetti Rosaria²,Barreca Maria Letizia³^ORCID,Ngo Liza⁴,Pescatori Luca¹^ORCID,Messore Antonella¹^ORCID,Pupo Giovanni¹^ORCID,Saccoliti Francesco¹^ORCID,Valente Sergio¹^ORCID,Mai Antonello¹^ORCID,Scipione Luigi¹^ORCID,Zheng Yujun George⁴^ORCID,Tintori Cristina⁵^ORCID,Botta Maurizio⁵^ORCID,Cecchetti Violetta³^ORCID,Altucci Lucia²⁶^ORCID,Di Santo Roberto¹^ORCID,Costi Roberta¹^ORCID

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti; “Sapienza” Università di Roma; P.le Aldo Moro 5 00185 Roma Italy

2. Dipartimento di Biochimica, Biofisica e Patologia generale; Università degli Studi della Campania Luigi Vanvitelli; Vico L. De Crecchio 7 80138 Napoli Italy

3. Department of Pharmaceutical Sciences; University of Perugia; Via A. Fabretti 48 06123 Perugia Italy

4. Department of Pharmaceutical and Biochemical Sciences; University of Georgia; Athens GA 30602 USA

5. Dipartimento di Biotecnologie, Chimica e Farmacia; Università degli Studi di Siena; Via Aldo Moro 2 53100 Siena Italy

6. Istituto di Genetica e Biofisica; IGB “Adriano Buzzati Traverso”; Via P. Castellino 111 80131 Napoli Italy

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201700040/fullpdf

Reference62 articles.

1. Molecular cloning and functional analysis of the adenovirus E1A-associated 300-kD protein (p300) reveals a protein with properties of a transcriptional adaptor.

2. Acetylation of Histones and Transcription-Related Factors

3. Epigenetic Regulation of the Latency-Associated Region of Marek's Disease Virus in Tumor-Derived T-Cell Lines and Primary Lymphoma

4. Histone Modification Pattern of the T-Cellular Herpesvirus Saimiri Genome in Latency

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