From Ergolines to Indoles: Improved Inhibitors of the Human H3 Receptor for the Treatment of Narcolepsy-Reference-Cited by-同舟云学术

From Ergolines to Indoles: Improved Inhibitors of the Human H3 Receptor for the Treatment of Narcolepsy

Published:2014-11-12 Issue:2 Volume:10 Page:266-275
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Auberson Yves P.,Troxler Thomas,Zhang Xuechun,Yang Charles R.,Feuerbach Dominik,Liu Yu-Chih,Lagu Bharat,Perrone Mark,Lei Lijun,Shen Xiaoxia,Zhang Dushan,Wang Chunxiu,Wang Tie-Lin,Briner Karin,Bock Mark G.

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Reference14 articles.

1. Histamine H3 Receptors and Sleep-Wake Regulation

2. Histamine H3 Antagonists as Wake-Promoting and Pro-Cognitive Agents

3. Cover Picture: Ergoline-Derived Inverse Agonists of the Human H3 Receptor for the Treatment of Narcolepsy (ChemMedChem 8/2014)

4. Correlation between ex Vivo Receptor Occupancy and Wake-Promoting Activity of Selective H3 Receptor Antagonists

5. Pharmacological Properties and Procognitive Effects of ABT-288, a Potent and Selective Histamine H3Receptor Antagonist

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