Design and Synthesis of Terephthalic Acid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Anti‐ Plasmodium Activity-Reference-Cited by-同舟云学术

Design and Synthesis of Terephthalic Acid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Anti‐ Plasmodium Activity

Published:2017-09-13 Issue:19 Volume:12 Page:1627-1636
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Stenzel Katharina¹²,Chua Ming Jang²,Duffy Sandra²,Antonova‐Koch Yevgeniya³,Meister Stephan³,Hamacher Alexandra¹,Kassack Matthias U.¹,Winzeler Elizabeth³,Avery Vicky M.²,Kurz Thomas¹,Andrews Katherine T.²,Hansen Finn K.¹⁴^ORCID

Affiliation:

1. Institute of Pharmaceutical and Medicinal Chemistry Heinrich Heine University Düsseldorf 40225 Düsseldorf Germany

2. Griffith Institute for Drug Discovery, Griffith University Don Young Road, Nathan Campus QLD 4111 Australia

3. Department of Pediatrics School of Medicine University of California, San Diego 9500 Gilman Drive 0741 La Jolla CA 92093 USA

4. Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy Leipzig University Brüderstraße 34 04103 Leipzig Germany

Funder

Deutscher Akademischer Austauschdienst

Deutsche Forschungsgemeinschaft

Australian Research Council

Medicines for Malaria Venture

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201700360

Reference61 articles.

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2. RTS S Clinical Trials Partnership The Lancet2015 386 31–45.

3. Sterile protection against human malaria by chemoattenuated PfSPZ vaccine

4. Malaria vaccine: WHO position paper—January 2016 The Weekly Epidemiological Record (WER) World Health Organization 2016 pp. 33–52;http://www.who.int/wer/2016/wer9104.pdf?ua=1(accessed September 5 2017).

5. Fighting drug-resistant Plasmodium falciparum: the challenge of artemisinin resistance

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