Potent HIV‐1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein‐Ligand X‐ray Structural Studies-Reference-Cited by-同舟云学术

Potent HIV‐1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein‐Ligand X‐ray Structural Studies

Published:2019-10-04 Issue:21 Volume:14 Page:1863-1872
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Ghosh Arun K.¹^ORCID,Xia Zilei¹,Kovela Satish¹,Robinson William L.¹,Johnson Megan E.¹,Kneller Daniel W.²,Wang Yuan‐Fang²,Aoki Manabu³⁴,Takamatsu Yuki⁴,Weber Irene T.²,Mitsuya Hiroaki⁵³⁴

Affiliation:

1. Department of Chemistry and Department of Medicinal Chemistry Purdue University West Lafayette IN 47907 USA

2. Departments of Biology and Chemistry, Molecular Basis of Disease Georgia State University Atlanta GA 30303 USA

3. Experimental Retrovirology Section, HIV and AIDS Malignancy Branch National Cancer Institute Bethesda MD 20892 USA

4. Department of Refractory Viral Infections National Center for Global Heath and Medicine Research Institute Shinjuku Tokyo 162-8655 Japan

5. Departments of Hematology and Infectious Diseases Kumamoto University School of Medicine Kumamoto 860-8556 Japan

Funder

National Institutes of Health

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201900508

Reference50 articles.

1. Structure-Based Design of Drugs and Other Bioactive Molecules

2. Structure-Based Drug Discovery

3. Recent Progress in the Development of HIV-1 Protease Inhibitors for the Treatment of HIV/AIDS

4. INHIBITORS OF HIV-1 PROTEASE: A Major Success of Structure-Assisted Drug Design

5. The development of antiretroviral therapy and its impact on the HIV-1/AIDS pandemic

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