Design, Synthesis, and Biological Evaluation of Tetrahydro-β-carboline Derivatives as Selective Sub-Nanomolar Gelatinase Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of Tetrahydro-β-carboline Derivatives as Selective Sub-Nanomolar Gelatinase Inhibitors

Published:2018-06-12 Issue:13 Volume:13 Page:1343-1352
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Mangiatordi Giuseppe Felice¹²,Guzzo Tatiana³,Rossano Eugenio Claudio³,Trisciuzzi Daniela¹,Alberga Domenico¹,Fasciglione Giovanni⁴,Coletta Massimiliano⁴,Topai Alessandra³,Nicolotti Orazio¹^ORCID

Affiliation:

1. Dipartimento di Farmacia-Scienze del Farmaco; Università di Bari “Aldo Moro”; Via Orabona, 4 70126 Bari Italy

2. Istituto Tumori IRCCS Giovanni Paolo II; Bari Italy

3. C4T S.r.l Colosseum Combinatorial Chemistry Centre for Technology; Via della Ricerca Scientifica snc, Ed. PP2-Macroarea Scienze 00133 Rome Italy

4. Dipartimento di Scienze cliniche e Medicina Traslazionale; Università di Roma “Tor Vergata”; Via Montpellier, 1 00133 Rome Italy

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201800237/fullpdf

Reference59 articles.

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