Inhibition of hypoxia-inducible transcription factor complex with designed epipolythiodiketopiperazine
Author:
Publisher
Wiley
Subject
Organic Chemistry,Biomaterials,Biochemistry,General Medicine,Biophysics
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1. Natural epidithiodiketopiperazine alkaloids as potential anticancer agents: Recent mechanisms of action, structural modification, and synthetic strategies;Bioorganic Chemistry;2023-08
2. Chetocochliodins A-I, Epipoly(thiodioxopiperazines) from Chaetomium cochliodes;Journal of Natural Products;2020-03-02
3. Inhibition of the HIF1α-p300 interaction by quinone- and indandione-mediated ejection of structural Zn(II);European Journal of Medicinal Chemistry;2015-04
4. Epidithiodiketopiperazines (ETPs) exhibit in vitro antiangiogenic and in vivo antitumor activity by disrupting the HIF-1α/p300 complex in a preclinical model of prostate cancer;Molecular Cancer;2014-04-28
5. Protein domain mimetics as in vivo modulators of hypoxia-inducible factor signaling;Proceedings of the National Academy of Sciences;2013-09-09
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