Cell‐Active, Reversible, and Irreversible Covalent Inhibitors That Selectively Target the Catalytic Lysine of BCR‐ABL Kinase-Reference-Cited by-同舟云学术

Cell‐Active, Reversible, and Irreversible Covalent Inhibitors That Selectively Target the Catalytic Lysine of BCR‐ABL Kinase

Published:2022-04-29 Issue:26 Volume:134 Page:
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angewandte Chemie

Author:

Chen Peng¹,Sun Jie¹,Zhu Chengjun²³,Tang Guanghui⁴,Wang Wei¹,Xu Manyi⁵,Xiang Menghua¹,Zhang Chong‐Jing⁵,Zhang Zhi‐Min²³,Gao Liqian¹,Yao Shao Q.⁴^ORCID

Affiliation:

1. School of Pharmaceutical Sciences (Shenzhen) Sun Yat-sen University Shenzhen 518107 China

2. School of Pharmacy Jinan University 601 Huangpu Avenue West Guangzhou 510632 China

3. Guangdong Youmei Institute of Intelligent Bio-manufacturing Foshan Guangdong 528200 China

4. Department of Chemistry National University of Singapore Singapore 117543 Singapore

5. State Key Laboratory of Bioactive Substances and Functions of Natural Medicines and Beijing Key Laboratory of Active Substances Discovery and Drugability Evaluation, Institute of Materia Medica, Peking Union Medical College and Chinese Academy of Medical Sciences Beijing 100050 China

Funder

National Natural Science Foundation of China

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.202203878

Reference62 articles.

1. Chronic myeloid leukemia: 2016 update on diagnosis, therapy, and monitoring

2. Past, present, and future of Bcr-Abl inhibitors: from chemical development to clinical efficacy

3. The resurgence of covalent drugs

4. Targeted Covalent Inhibitors for Drug Design

5. Zielgerichtete kovalente Inhibitoren für das Wirkstoffdesign

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3. RGD Cyclopeptide Equipped with a Lysine‐Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency;Chemistry – A European Journal;2023-02-27