Discovery of a Potent Degrader for Fibroblast Growth Factor Receptor 1/2-Reference-Cited by-同舟云学术

Discovery of a Potent Degrader for Fibroblast Growth Factor Receptor 1/2

Published:2021-06-14 Issue:29 Volume:133 Page:16041-16047
ISSN:0044-8249
Container-title:Angewandte Chemie
language:en
Short-container-title:Angew. Chem.

Author:

Du Guangyan¹²,Jiang Jie¹²,Wu Qibiao³⁴,Henning Nathaniel J.¹²,Donovan Katherine A.¹²,Yue Hong¹²,Che Jianwei¹²,Lu Wenchao¹²,Fischer Eric S.¹²,Bardeesy Nabeel³⁴,Zhang Tinghu⁵,Gray Nathanael S.⁵^ORCID

Affiliation:

1. Department of Cancer Biology Dana Farber Cancer Institute 360 Longwood Ave Boston MA 02215 USA

2. Department of Biological Chemistry and Molecular Pharmacology Harvard Medical School Boston MA USA

3. Cancer Center Massachusetts General Hospital Harvard Medical School Boston MA USA

4. Broad Institute of Harvard and MIT Cambridge MA USA

5. Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine Stanford University Stanford CA USA

Funder

National Institutes of Health

Pediatric Low Grade Astrocytoma Foundation

V Foundation for Cancer Research

Cholangiocarcinoma Foundation

Publisher

Wiley

Subject

General Medicine

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.202101328

Reference56 articles.

1. The FGF family: biology, pathophysiology and therapy

3. Inhibition of the fibroblast growth factor receptor (FGFR) pathway: the current landscape and barriers to clinical application

4. Structure, activation and dysregulation of fibroblast growth factor receptor kinases: perspectives for clinical targeting

5. Fibroblast growth factor receptors as treatment targets in clinical oncology

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