Synthetic Approaches Used in the Scale-Up of Macrocyclic Clinical Candidates
Author:
Affiliation:
1. Department of Process Research & Development, Merck Research Laboratories; Merck & Co., Inc.; Rahway NJ USA
Publisher
John Wiley & Sons, Inc.
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1002/9781119092599.ch15/fullpdf
Reference69 articles.
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2. Macrocyclic drugs and synthetic methodologies toward macrocycles;Yu;Molecules,2013
3. How beyond rule of 5 drugs and clinical candidates bind to their targets;Doak;J. Med. Chem.,2016
4. Macrocycles in new drug discovery;Mallinson;Future Med. Chem.,2012
5. Macrocyclic drugs and clinical candidates: what can medicinal chemists learn from their properties?;Giordanetto;J. Med. Chem.,2014
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